Lebitso la lebitso | ActiTide-AH3 |
Nomoro ea CAS. | 616204-22-9 |
INCI Lebitso | Acetyl Hexapeptide-8 |
Kopo | Lotion, Serum, Mask, Sehloekisi sa sefahleho |
Sephutheloana | 100g / botlolo, 1kg / mokotla |
Ponahalo | Phofo e tšoeu ho isa ho e tšoeu |
Solubility | Metsi a qhibilihang |
Mosebetsi | Letoto la li-peptide |
Shelf bophelo | lilemo tse 2 |
Polokelo | Boloka setshelo se koetsoe ka thata sebakeng se phodileng, se omeletseng ho 2 - 8°C. |
Tekanyetso | 0.005-0.05% |
Kopo
Lipatlisiso tse mabapi le mekhoa ea mantlha e thibelang wrinkles li lebisitse ho sibolloeng ha ActiTide-AH3, e leng hexapeptide e ncha e ntlafalitsoeng ka mokhoa oa mahlale ho tloha ho moralo o hlakileng ho isa tlhahiso ea GMP, ka litholoana tse ntle.
ActiTide-AH3 e fana ka katleho ea ho fokotsa mats'oenyeho e bapisoang le Mofuta oa A oa Chefo ea Botulinum, ha e ntse e qoba likotsi tsa ente le ho fana ka katleho e kholo ea litšenyehelo.
Melemo ea Litlolo:
ActiTide-AH3 e fokotsa botebo bo sosobaneng bo bakoang ke ho honyela ha mesifa ea sefahleho, ka litlamorao tse hlahelletseng phatleng le makukuno a periocular.
Mokhoa oa ts'ebetso:
Ho honyela ha mesifa ho etsahala ha li-neurotransmitter li lokolloa li-synaptic vesicles. The SNARE complex - kopano ea ternary ea VAMP, Syntaxin, le SNAP-25 protheine - ke ea bohlokoa bakeng sa vesicle docking le neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). E rarahaneng ena e sebetsa e le hook ea cellular, e hapang li-vesicles le ho khanna membrane fusion.
Joalo ka sebopeho sa sebopeho sa SNAP-25 N-terminus, ActiTide-AH3 e qothisana lehlokoa le SNAP-25 bakeng sa ho kengoa setsing sa SNARE, ho hlophisa kopano ea eona. Ho senyeha ha SNARE complex ho sitisa vesicle docking le ho lokolloa ha li-neurotransmitter, ho lebisang ho fokotseheng ha mesifa le ho thibela ho sosobana le ho thehoa ha mela e metle.
ActiTide-AH3 ke mokhoa o sireletsehileng haholoanyane, oa moruo, hape o bonolo ho fapana le Botulinum Toxin Type A. E shebane haholo le tsela e ts'oanang ea ho etsa matsutsuba empa e sebetsa ka mokhoa o ikhethileng.