Lebitso la lebitso | ActiTide-AH3(Liquefied 500) |
Nomoro ea CAS. | 7732-18-5; 616204-22-9; 1117-86-8 |
INCI Lebitso | Metsi; Acetyl hexapeptide-8; Caprylyl glycol |
Kopo | Lotion, Serum, Mask, Sehloeki sa sefahleho |
Sephutheloana | 1kg/botlolo |
Ponahalo | Mokelikeli o hlakileng le o bonaletsang |
Likahare tsa Peptide | 0.045 - 0.060% |
Solubility | Metsi a qhibilihang |
Mosebetsi | Letoto la li-peptide |
Shelf bophelo | lilemo tse 2 |
Polokelo | Boloka sebakeng se phodileng le se omileng, hole le leseli. 2 ~ 8°C bakeng sa polokelo |
Tekanyetso | 3.0-10.0% |
Kopo
Lipatlisiso tse mabapi le mekhoa ea mantlha e thibelang wrinkles li lebisitse ho sibolloeng ha ActiTide-AH3, e leng hexapeptide e ncha e ntlafalitsoeng ka mokhoa oa mahlale ho tloha ho moralo o hlakileng ho isa tlhahiso ea GMP, ka litholoana tse ntle.
ActiTide-AH3 e fana ka katleho ea ho fokotsa mats'oenyeho e bapisoang le Mofuta oa A oa Chefo ea Botulinum, ha e ntse e qoba likotsi tsa ente le ho fana ka katleho e kholo ea litšenyehelo.
Melemo ea Litlolo:
ActiTide-AH3 e fokotsa botebo bo sosobane bo bakoang ke ho honyela ha mesifa ea sefahleho, ka litlamorao tse hlahelletseng phatleng le makukuno a periocular.
Mokhoa oa ts'ebetso:
Ho honyela ha mesifa ho etsahala ha li-neurotransmitter li lokolloa li-synaptic vesicles. The SNARE complex - kopano ea ternary ea VAMP, Syntaxin, le SNAP-25 protheine - ke ea bohlokoa bakeng sa vesicle docking le neurotransmitter exocytosis (A. Ferrer Montiel et al., JBC 1997, 272: 2634-2638). E rarahaneng ena e sebetsa e le hook ea cellular, e hapang li-vesicles le ho khanna membrane fusion.
Joalo ka sebopeho sa sebopeho sa SNAP-25 N-terminus, ActiTide-AH3 e qothisana lehlokoa le SNAP-25 bakeng sa ho kengoa setsing sa SNARE, ho hlophisa kopano ea eona. Ho senyeha ha SNARE complex ho sitisa vesicle docking le ho lokolloa ha li-neurotransmitter, ho lebisang ho fokotseheng ha mesifa le ho thibela ho sosobana le ho thehoa ha mela e metle.
ActiTide-AH3 ke mokhoa o sireletsehileng haholoanyane, oa moruo, hape o bonolo ho fapana le Botulinum Toxin Type A. E shebane haholo le tsela e ts'oanang ea ho etsa matsutsuba empa e sebetsa ka mokhoa o ikhethileng.